PQ401
- PQ 401
货号: abs813318
货号-规格 | 货期 | 价格 | 数量 |
abs813318-5mg | 1-2周 | ¥759.00 | - + |
abs813318-10mg | 1-2周 | ¥972.00 | - + |
abs813318-25mg | 1-2周 | ¥1766.00 | - + |
abs813318-50mg | 1-2周 | ¥3063.00 | - + |

产品描述 | |
描述 | PQ 401抑制IGF-1R区域自磷酸化,IC50为低于1 μM。PQ 401是IGF-1R 抑制剂,浓度<100 nM时,抑制IGF-IR激酶域的自磷酸化,IC50 < 1μM. PQ 401显著降低MCF-7细胞增殖,IC50为8 μM。PQ 401也抑制MCNeuA细胞生长,IC50为15 μM。PQ 401作用于MCF-7 细胞,抑制IGF-I调节的抗凋亡途径。 |
纯度 | >98% |
储存/保存方法 | Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. |
基本信息 | |
别名 | PQ 401 |
可溶性/溶解性 | Ethanol :8.5 mg/mL (25 mM) DMSO :17.1 mg/mL (50 mM) |
生物活性 | |
靶点 | IGF-1R |
In vitro(体外研究) | PQ 401 is an IGF-1R inhibitor and inhibits autophosphorylation of the IGF-IR kinase domain at concentrations |
In vivo(体内研究) | PQ 401 (50 mg/Kg, 100 mg/Kg) significantly inhibits MCNeuA tumor growth in a dose-dependent manner. |
参考文献 | |
参考文献 |