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  • Sumanirole Maleate
    • U95666E; PNU 95666; PNU 95666E; Sumanirole
    货号: abs813950
    CAS号: 179386-44-8
    分子式: C11H13N3O.C4H4O4
    分子量: 319.31
    产品说明书
    分享:
    货号-规格 货期 价格 数量
    abs813950-5mg 1-2周 ¥1067.00
    - +
    abs813950-10mg 1-2周 ¥1742.00
    - +
    abs813950-25mg 1-2周 ¥3881.00
    - +
    abs813950-50mg 1-2周 ¥6549.00
    - +
    大包装询价
    产品描述
    描述

    Sumanirole maleate is a highly selective D2 receptor full agonist with an ED50 of about 46 nM. It has greater than 200-fold selectivity for the D2 receptor subtype versus the other dopamine receptor subtypes in radioligand binding assays. In cell-based assays, sumanirole is a fully efficacious agonist, with EC50 values between 17 and 75 nM. In animals, sumanirole elicits many physiological responses attributed to D2-like receptor function. In rats, sumanirole is a full agonist for elevation of striatal acetylcholine levels (ED50 = 12.1 μmol/kg i.p.). Sumanirole s.c. dose dependently decreased plasma prolactin levels and depressed dopamine neuron firing rates in the substantia nigra pars compacta with an ED50 of 2.3 μmol/kg i.v.

    纯度
    >98%
    储存/保存方法
    store at -20℃ for one year(Powder);
    in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months.
    基本信息
    别名
    U95666E; PNU 95666; PNU 95666E; Sumanirole
    外观
    白色货类白色粉末
    可溶性/溶解性
    10 mM in DMSO
    温馨提示:本产品仅作科研实验使用,不支持临床等研究
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