Cangrelor Tetrasodium
- 坎格雷洛四钠盐;AR-C69931MX;AR-C69931
货号: abs814683
货号-规格 | 货期 | 价格 | 数量 |
abs814683-5mg | 1-2周 | ¥992.00 | - + |
abs814683-25mg | 1-2周 | ¥3087.00 | - + |

产品描述 | |
描述 | Cangrelor is a potent, competitive P2Y12 receptor inhibitor that is administered by intravenous infusion and rapidly achieves near complete inhibition of ADP-induced platelet aggregation. |
纯度 | 98% |
储存/保存方法 | Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. |
基本信息 | |
别名 | 坎格雷洛四钠盐;AR-C69931MX;AR-C69931 |
外观 | powder |
可溶性/溶解性 | DMSO :2 mg/mL (2.31 mM) Water :100 mg/mL (115.70 mM) |
生物活性 | |
靶点 | P2Y12 receptor |
In vitro(体外研究) | Cangrelor is an intravenous ATP analog that directly inhibits, without the need for being metabolized, the P2Y12 receptor in a reversible manner. Cangrelor has a rapid-onset and -offset mechanism of action and achieves significantly greater degrees of platelet inhibition compared with clopidogrel. |
In vivo(体内研究) | Cangrelor is rapidly deactivated by plasmatic ectonucleotidases and, thus, has an extrmely short half-life (2-5 min). Preclinical studies performed in animal models in the early stages of cangrelor development show efficacy in inhibiting thrombus formation and ADP-induced platelet aggregation, as well as a lower increase of bleeding times when compared with IIb/IIIa antagonist. |
温馨提示:本产品仅作科研实验使用,不支持临床等研究 |
- 实验方法 实验条件
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