17 alpha-propionate
- 克拉司酮;Clascoterone;CB-03-01;Cortexolone 17α-propionate;Cortexolone 17 alpha-propionate
货号: abs811002
货号-规格 | 货期 | 价格 | 数量 |
abs811002-50mg | 1-2周 | ¥1250.00 | - + |
abs811002-100mg | 1-2周 | ¥1750.00 | - + |
abs811002-500mg | 1-2周 | ¥5250.00 | - + |

产品描述 | ||
描述 | 17 alpha-propionate is a new topical and peripherally selective androgen antagonist. | |
纯度 | >98% | |
储存/保存方法 | Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. | |
基本信息 | ||
别名 | 克拉司酮;Clascoterone;CB-03-01;Cortexolone 17α-propionate;Cortexolone 17 alpha-propionate | |
外观 | White to off white powder | |
可溶性/溶解性 | DMSO : ≥ 100 mg/mL (248.43 mM) | |
生物活性 | ||
靶点 | Androgen Receptor | |
In vivo(体内研究) | Clascoterone is a new potent topical antiandrogen potentially useful in acne vulgaris. Clascoterone 1% cream was very well tolerated, and was significantly better than placebo regarding TLC (P = 0·0017), ILC (P = 0·0134) and ASI (P = 0·0090), and also clinically more effective than comparator. The product also induced a faster attainment of 50% improvement in all the above parameters. | |
温馨提示:本产品仅作科研实验使用,不支持临床等研究 |
- 实验方法 实验条件
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